海绵Mycale adhaerens 13-deoxytedanolide IC50为9.5×10-5mg·ml-1,T/C=189%
茜草Rubia cordifolia 环已肽,RA-Ⅷ,RA-Ⅻ IC50<0.05mg·ml-1
海绵 theonella sp. Keramamide F, orbiculamide A, theonella peptolides Ia~Ie L1210强活性,IC50 1.4~2.4mg·ml-1
加勒比海海绵Discordemia sp. polydiscamide A A549IC50< 0.7mg·ml-1
海鞘Diazona chinensis diazonamides A, B HCT-116和B16 IC50<0.015mg·ml-1
海绵 stylotella auranticum Stylostatin I ED50 0.8mg·ml-1
海鞘 Trididemnum solidum didemnin B(X,Y) Ⅱ期临床
印度洋海鞘 Lissodinum patclla Ulithiaclamide B KBcell ID50 17ng/ml-1
紫杉醇 Taxus sp. 紫杉烷类二萜 Taxol 抗癌谱广泛,干扰微管蛋白
雷公藤Tripterygium sp. triptolid(1),tripdiolide(2), triptonide(3) (1),(2)对LE、PS有效剂量为0.1mg/kg
